I-N-Boc-Glycine Isoproploplopy

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I-N-Boc-Glycine Isoproploplopy

Umzi mveliso wamayeza uxhomekeke kakhulu kwiikominyi zekhemikhali zokuphuhlisa amayeza asebenzayo nawo akhuselekileyo. Enye enjalo efumene ingqalelo enkulu yileN-boc-vlycine pooproplopyter. Le michiza iguquguqukayo idlala indima ebalulekileyo kwiSingqutyha yemveliso eyahlukeneyo yamayeza, ihambisa iipropathi ezahlukileyo ezikhuthaza iinkqubo zophuhliso lweziyobisi. Kweli nqaku, siza kuphonononga izicelo zamayeza ze-N-Blycine ye-Isoproploploplopysine kwaye kutheni liyinxalenye ebalulekileyo kulowo.

Yintoni i-n-boc-vlycine pooproploplopleter?
I-N-Blycine ye-Isoproploploploperter yifom eguqulweyo ye-gelycine, i-amino acid esebenza njengebhlokhi yesakhiwo. Iqela "N-Boc-ButoXycarbol) kunye ne-IyopipyCl kunye ne-Iyopropyl Derter Amaqela okhulisa amaqela akhuselayo aphucula uzinzo lwequmrhu kunye nokukhulisa kwakhona. Oku kwenza i-N-Blycine yase-Isoproplopyter ixabisekileyo ephakathi kwiSynthesic Synthesi, ngakumbi kumzi-mveliso wamachiza.

Izicelo eziphambili zamayeza ezi-zuza ze-N-Blycine Isoproplopyter
I-1. I-Peptide Synthesis
Olunye losetyenziso oluphambili lwe-N-Blycine ye-Isoproploplopleter kwi-Syntheside ye-Peptrade. I-peptides ziikhonkco ezimfutshane zee-Amino Acids ezidlala indima ebalulekileyo kwiinkqubo zebhayoloji kwaye zisenziwa njengeearhente zonyango. Iqela le-N-B-BoC likhusela iqela le-Amino ngexesha leSynthesis, ngelixa iSopropyl Esterl iququzelele ukumiswa kweebhondi zepeptide. Oku kwenza i-N-Blycine ye-Isoproploplopleter inyanzelekile i-regent eyimfuneko yokuvelisa i-peptides ngobunyulu obuphezulu kunye nesivuno.
2. Iziyobisi eziphakathi
I-N-Boc-Glycine Isoproploploploperser isetyenziswe ngokubanzi njengendawo ephakathi kwi-synthesical yezinto ezahlukeneyo zamayeza. Amaqela ayo okhuselayo avumela oosomamichiza ukuba benze izinto ezikhethiweyo zokukhetha, besenza ukuba kubekho ukudalwa kweemolekyuli ezintsonkothileyo. Oku kubaluleke kakhulu ekuphuhlisweni kweentsholongwane, ii-antivirals, kunye neziyobisi ezintiyo.
3. Uphuhliso lwe-rodrug
I-Prodrugs ziindawo ezingasebenziyo eziguqulayo ziguqula ichiza elisebenzayo ngaphakathi komzimba. Iqela le-Iyopropyl Ester kwi-N-Blycine Isoproploplopyter inokusetyenziselwa ukuyila i-prodrugs ephucula ukuhanjiswa kweziyobisi kunye nebhayili. Oku kuluncedo ngakumbi kumayeza afuna ukudlula inkqubo yokugaya ukutya okanye amaziko athile ajolise kuyo.
4. I-Enzyme ethi
I-Enzyme ethi i-Enzyme i-Enzyme ikwiklasi yeziyobisi ezithintela umsebenzi wee-enzymes ezithile, zihlala zidla ngokunyanga izifo ezinjengomhlaza kunye nosulelo lwentsholongwane. I-N-Blycine Isoproploplopleter isebenza njengebhloko yesakhiwo yokudibanisa ezi zinto zithintelayo, ngenxa yokwazi kwako ukuchaza ezizinzileyo nezingasebenziyo.
I-5. Isiseko sekhemikhali sekhemikhali
Ukugxila kwe-N-Blycine ye-Isoproploplopyter kwenza isixhobo esibalulekileyo seSynthesic Synthesic. Abaphandi bamayeza bayisebenzisa ukwenza i-inovels comples ezinefuthe lonyango, ukukhawulezisa ukufunyanwa kwamachiza amatsha.

Izibonelelo zokusebenzisa i-N-Blycine ye-Isoproploploplester kwi-Hermaceuticals
Ukusetyenziswa kwe-N-Blycine ye-Isoproploplopleter kwi-STIPROCENCE kwi-STIPROCENTIONS kwi-STIPRORDE inikezela izibonelelo ezininzi:
Ukuhlaziywa okuphezulu: Amaqela okhuselo aphucule i-compountical yendawo, evumela ukwenziwa ngokufanelekileyo kwezifo zemolekyuli ezinzima.
• Uzinzo: Iqela le-N-B-Boc libonelela ngozinzo ngexesha lokuphendula kwemichiza, ukunciphisa umngcipheko wokuphendula esecaleni okungafunekiyo.
• Ukusetyenziswa gwenxa: Izicelo zayo zisusela kwi-Syntheside yoPhuculo, esenza isixhobo esiguquguqukayo kubaphandi.
• I-Sciallifcy: I-N-Boc-Glycine Isoproploplopyter ilungele uphando oluncinci lwelebhu kunye nemveliso enkulu yeshishini.

Imiceli mngeni kunye nokuqwalaselwa
Ngelixa i-N-Blycine ye-Isoproplopyter inikezela ngezibonelelo ezininzi, ukusetyenziswa kwayo kwiindawo zamayeza nazo kuza nemiceli mngeni. Umzekelo, ukususwa kweqela lokukhusela i-N-Boc kufuna iimeko ezithile, ekufuneka zilawulwa ngononophelo ukuthintela ukonakalisa imveliso yokugqibela. Ukongeza, iindleko ze-charty n-boc-vlycine pooproploplopleter zinokuqwalaselwa kwizicelo ezininzi.
Ngaphandle kolu celomngeni, uphando oluqhubekayo kunye nokuhambela phambili kwezobuchwephesha kunye nokwenza le micimbi, ukwenza i-N-Boc-Glycine Isoproploploploplopleter ifikeleleke kwaye iqhubekeke ekuphuhlisweni kwe-farmaceutical.

Ikamva le-N-Blycine Isoproploplopy
Njengoko imfuno yamayeza enobuchule kunye nempumelelo iyaqhubeka ukhula, indima ye-N-Blycine Isoproploploplopy yophuhliso lweziyobisi kulindeleke ukuba yandise. Inkqubela phambili kwiChemistry yeSynthetic kunye nenkqubo yokusebenza kunokwenzeka ukomeleza izicelo zayo, ngakumbi kumacandelo amayeza abhalwe ngobuntu kunye neebhayilojini.
Ngapha koko, ukugxila okukhulayo kwi-chemistry eluhlaza kuqhuba uphuhliso lweendlela ezizinzileyo zokuyifumana kunye nokusebenzisa i-N-Glycine ye-iOproploploploplopy. Oku kulungelelaniswa nokukuzibophelela kweshishini le-chithaction ukunciphisa ifuthe lendalo esingqongileyo ngelixa sihambisa unyango olusindisa ubomi.

Ukuqukumbela
I-N-Boc-vlycine ye-Isoproploplopleter yindawo ebalulekileyo kumzi-mveliso wamachiza, kunye nezicelo ezisusela kwi-Syntheis yePeptima yoPhuculo. Iipropathi zayo ezahlukileyo, kubandakanya ukuvela okuphakathi kunye nokuzinza, zenze isixhobo esingazilekanga kubaphandi kunye nabavelisi ngokufanayo. Njengoko eli shishini liyaqhubeka nokulingisa, ukubaluleka kwe-N-Blycine ye-Isoproploplopy kwi-STIPROPERS kwi-STIPROPLESE kuphuhliso lwamachiza kusetwa ukukhulisa, ukuvula indlela yezisombululo ezitsha neziphuculweyo zonyango neziphuculweyo.
Ukuba ubandakanyeka kuphando lwamayeza okanye ukuveliswa, ukuqonda izicelo kunye nezibonelelo ze-N-Glycine Isoproploploploplester inokukunceda ukuba uqhubeke nokuphuhliswa kwamayeza e-gesing. Jonga ukuba le lelona qangalela iguquguqukayo linokuphucula njani umsebenzi wakho kunye nokuqhuba izinto ezintsha kwintsimi yamayeza.

Ukufumana ezinye iingcebiso kunye neengcali zengcali, ndwendwela iwebhusayithi yethuhttps: //wwwchem.net/Ukuze ufunde ngakumbi malunga neemveliso zethu kunye nezisombululo.


Ixesha lokuphumla: Mar-17 ukuya ku-525